Rational Design of Dual-Domain Binding Inhibitors for N-Acetylgalactosamine Transferase 2 with Improved Selectivity over the T1 and T3 Isoforms

Compañón, Ismael Ballard, Collin J. Lira-Navarrete, Erandi Santos, Tanausú Monaco, Serena Muñoz-García, Juan C. Delso, Ignacio Angulo, Jesus Gerken, Thomas A. Schjoldager, Katrine T. Clausen, Henrik Tejero, Tomás Merino, Pedro Corzana, Francisco Hurtado-Guerrero, Ramon Ghirardello, Mattia Rational Design of Dual-Domain Binding Inhibitors for N-Acetylgalactosamine Transferase 2 with Improved Selectivity over the T1 and T3 Isoforms

10.1021/jacsau.4c00633 2024

2024